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Trifluoperazine HCL /Maleate CAS NO.440-17-5
- FOB Price: USD: 1.00-1.00 /Kilogram Get Latest Price
- Min.Order: 1 Kilogram
- Payment Terms: L/C,D/A,D/P,T/T
- Available Specifications:
99%(1-500)Kilogram
- Product Details
Keywords
- 440-17-5
- Trifluoperazine hydrochloride
- Trifluoperazine dihydrochloride
Quick Details
- ProName: Trifluoperazine HCL /Maleate
- CasNo: 440-17-5
- Molecular Formula: C21H25ClF3N3S
- Appearance: white to pale yellow crystalline powd...
- Application: Central Nervous System Drug; Anti-Emet...
- DeliveryTime: prompt shipment
- PackAge: 25kg drum
- Port: Shanghai,China
- ProductionCapacity: 200 Metric Ton/Year
- Purity: 99%min
- Storage: sealed and stored in cool places.
- Transportation: BY SEA,AIR
- LimitNum: 1 Kilogram
- Related Substances: not avaliable
- Residue on Ignition: 0.1%
- Heavy Metal: ≤10ppm
- Valid Period: 2 years
- EINECS No: 207-123-0
Superiority
Trifluoperazine dihydrochloride
Trifluoperazine Dihydrochloride is a cell-permeable phenothiazine compound with antiadrenergic effects. Trifluoperazine is described as an antagonist of adrenergic receptors, demonstrating much higher activity at the α-1 over the α-2 adrenergic receptor. Trifluoperazine is also described to produce antidopaminergic effects. Trifluoperazine facilitates agonist induced elevation of cytosolic calcium at low concentrations (10μM), and antagonizes CaM (calmodulin) at higher concentrations. Potent and irreversible inhibitor of cAMP-gated cationic channels. Inhibits DNA repair. Potent neurotoxin. Trifluoperazine is an inhibitor of D2DR.
Details
guarantee the quality of Trifluoperazine dihydrochloride
|
Item |
Requirements |
Test Results |
|
Description |
A white to pale yellow crystalline powder Hygroscopic, freely soluble in water, soluble in alcohol |
Complies |
|
Identification |
A,B,C,D,E |
Complies |
|
Appearance of solution |
It is clear and colourless |
Complies |
|
Melting point |
About 242℃, with decomposition |
Complies |
|
Acidity |
1.6~2.5 |
2.0 |
|
Related substances |
Examine by thin-layer chromatography, using a TLC silica gel GF254 Plate R with a concentration zone. Not more than 0.5 percent |
Complies |
|
Sulphated ash |
≤0.10% |
0.05% |
|
Loss on drying |
≤1.5% |
0.43% |
|
Heavy Metal |
≤10ppm |
Complies |
|
Assay |
99.0%~101.0% |
99.6% |
|
Conclusion |
Meets the Requirement |
|